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P-Rex1 limits the agonist-induced internalization of GPCRs independently of its Rac-GEF activity

P-Rex1 activates Rac downstream of GPCRs to regulate processes ranging from innate immunity to neuronal plasticity, its deregulation contributing to cancer. Here, Baker et al. show that P-Rex1 also controls GPCR trafficking, limiting agonist-induced GPCR internalization through an adapter function. Thus, P-Rex1 promotes GPCR responses in a dual manner.

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